beta-cyclodextrin/epoxysuccinyl peptide conjugates: new drug targeting system for tumor cells

Schaschke, Norbert; Assfalg-Machleidt, I; Machleidt, W; Lassleben, T; Sommerhoff, CP; Moroder, L

beta-cyclodextrin/epoxysuccinyl peptide conjugates: new drug targeting system for tumor cells

Schaschke N, Assfalg-Machleidt I, Machleidt W, Lassleben T, Sommerhoff CP, Moroder L (2000)
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 10(7): 677-680.

Zeitschriftenaufsatz | Veröffentlicht | Englisch

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DOI

https://doi.org/10.1016/S0960-894X(00)00078-0

Autor*in

Schaschke, Norbert^UniBi; Assfalg-Machleidt, I; Machleidt, W; Lassleben, T; Sommerhoff, CP; Moroder, L

Einrichtung

Fakultät für Chemie > Organische Chemie III

Erscheinungsjahr

2000

Zeitschriftentitel

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Band

10

Ausgabe

7

Seite(n)

677-680

ISSN

0960-894X

Page URI

https://pub.uni-bielefeld.de/record/2403852

Zitieren

Schaschke N, Assfalg-Machleidt I, Machleidt W, Lassleben T, Sommerhoff CP, Moroder L. beta-cyclodextrin/epoxysuccinyl peptide conjugates: new drug targeting system for tumor cells. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 2000;10(7):677-680.

Schaschke, N., Assfalg-Machleidt, I., Machleidt, W., Lassleben, T., Sommerhoff, C. P., & Moroder, L. (2000). beta-cyclodextrin/epoxysuccinyl peptide conjugates: new drug targeting system for tumor cells. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 10(7), 677-680. https://doi.org/10.1016/S0960-894X(00)00078-0

Schaschke, Norbert, Assfalg-Machleidt, I, Machleidt, W, Lassleben, T, Sommerhoff, CP, and Moroder, L. 2000. “beta-cyclodextrin/epoxysuccinyl peptide conjugates: new drug targeting system for tumor cells”. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 10 (7): 677-680.

Schaschke, N., Assfalg-Machleidt, I., Machleidt, W., Lassleben, T., Sommerhoff, C. P., and Moroder, L. (2000). beta-cyclodextrin/epoxysuccinyl peptide conjugates: new drug targeting system for tumor cells. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 10, 677-680.

Schaschke, N., et al., 2000. beta-cyclodextrin/epoxysuccinyl peptide conjugates: new drug targeting system for tumor cells. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 10(7), p 677-680.

N. Schaschke, et al., “beta-cyclodextrin/epoxysuccinyl peptide conjugates: new drug targeting system for tumor cells”, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 10, 2000, pp. 677-680.

Schaschke, N., Assfalg-Machleidt, I., Machleidt, W., Lassleben, T., Sommerhoff, C.P., Moroder, L.: beta-cyclodextrin/epoxysuccinyl peptide conjugates: new drug targeting system for tumor cells. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 10, 677-680 (2000).

Schaschke, Norbert, Assfalg-Machleidt, I, Machleidt, W, Lassleben, T, Sommerhoff, CP, and Moroder, L. “beta-cyclodextrin/epoxysuccinyl peptide conjugates: new drug targeting system for tumor cells”. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 10.7 (2000): 677-680.

14 Zitationen in Europe PMC

Daten bereitgestellt von Europe PubMed Central.

Highly Functionalized β-Cyclodextrins by Solid-Supported Synthesis.
Vurgun N, Nitz M., Chemistry 24(17), 2018
PMID: 29389050

On the synthesis of cyclodextrin-peptide conjugates by the Huisgen reaction.
Lartia R, Jankowski CK, Arseneau S., J Pept Sci 22(8), 2016
PMID: 27443976

Cyclodextrin-peptide conjugates for sequence specific DNA binding.
Ruiz García Y, Zelenka J, Pabon YV, Iyer A, Buděšínský M, Kraus T, Smith CI, Madder A., Org Biomol Chem 13(18), 2015
PMID: 25857557

New glycoside derivatives of carnosine and analogs resistant to carnosinase hydrolysis: synthesis and characterization of their copper(II) complexes.
Lanza V, Bellia F, D'Agata R, Grasso G, Rizzarelli E, Vecchio G., J Inorg Biochem 105(2), 2011
PMID: 21194616

Click synthesis of estradiol-cyclodextrin conjugates as cell compartment selective estrogens.
Kim HY, Sohn J, Wijewickrama GT, Edirisinghe P, Gherezghiher T, Hemachandra M, Lu PY, Chandrasena RE, Molloy ME, Tonetti DA, Thatcher GR., Bioorg Med Chem 18(2), 2010
PMID: 20031420

Synthesis and pharmacological evaluation of a new targeted drug carrier system: beta-cyclodextrin coupled to oxytocin.
Bertolla C, Rolin S, Evrard B, Pochet L, Masereel B., Bioorg Med Chem Lett 18(6), 2008
PMID: 18296049

Cyclodextrin/imatinib complexation: binding mode and charge dependent stabilities.
Béni S, Szakács Z, Csernák O, Barcza L, Noszál B., Eur J Pharm Sci 30(2), 2007
PMID: 17145172

Analysis of carbohydrates and glycoconjugates by matrix-assisted laser desorption/ionization mass spectrometry: An update covering the period 1999-2000.
Harvey DJ., Mass Spectrom Rev 25(4), 2006
PMID: 16642463

Solid-phase synthesis of double-headed epoxysuccinyl activity-based probes for selective targeting of papain family cysteine proteases.
Verhelst SH, Bogyo M., Chembiochem 6(5), 2005
PMID: 15776409

Crystal structure of NS-134 in complex with bovine cathepsin B: a two-headed epoxysuccinyl inhibitor extends along the entire active-site cleft.
Stern I, Schaschke N, Moroder L, Turk D., Biochem J 381(pt 2), 2004
PMID: 15084146

1,2,4-thiadiazole: a novel Cathepsin B inhibitor.
Leung-Toung R, Wodzinska J, Li W, Lowrie J, Kukreja R, Desilets D, Karimian K, Tam TF., Bioorg Med Chem 11(24), 2003
PMID: 14642597

Epoxysuccinyl peptide-derived cathepsin B inhibitors: modulating membrane permeability by conjugation with the C-terminal heptapeptide segment of penetratin.
Schaschke N, Deluca D, Assfalg-Machleidt I, Höhneke C, Sommerhoff CP, Machleidt W., Biol Chem 383(5), 2002
PMID: 12108551

Bivalent inhibition of human beta-tryptase.
Schaschke N, Matschiner G, Zettl F, Marquardt U, Bergner A, Bode W, Sommerhoff CP, Moroder L., Chem Biol 8(4), 2001
PMID: 11325588

Epoxysuccinyl peptide-derived affinity labels for cathepsin B.
Schaschke N, Assfalg-Machleidt I, Lassleben T, Sommerhoff CP, Moroder L, Machleidt W., FEBS Lett 482(1-2), 2000
PMID: 11018529

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