Upgrading a Natural Product: Inhibition of Human beta-Tryptase by Cyclotheonamide Analogues

Schaschke N, Sommerhoff CP (2010)
CHEMMEDCHEM 5(3): 367-370.

Zeitschriftenaufsatz | Veröffentlicht | Englisch
 
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DOI
Autor*in
Schaschke, NorbertUniBi; Sommerhoff, Christian P.
Einrichtung
Centrum für Biotechnologie > Arbeitsgruppe N. Schaschke
Fakultät für Chemie > Organische Chemie III
Centrum für Biotechnologie > Institut für Biochemie und Biotechnik
Stichworte
proteases; relationships; mast cells; beta-amino acids; peptides; structure-activity
Erscheinungsjahr
2010
Zeitschriftentitel
CHEMMEDCHEM
Band
5
Ausgabe
3
Seite(n)
367-370
ISSN
1860-7179
eISSN
1860-7187
Page URI
https://pub.uni-bielefeld.de/record/2403708

Zitieren

Schaschke N, Sommerhoff CP. Upgrading a Natural Product: Inhibition of Human beta-Tryptase by Cyclotheonamide Analogues. CHEMMEDCHEM. 2010;5(3):367-370.
Schaschke, N., & Sommerhoff, C. P. (2010). Upgrading a Natural Product: Inhibition of Human beta-Tryptase by Cyclotheonamide Analogues. CHEMMEDCHEM, 5(3), 367-370. https://doi.org/10.1002/cmdc.200900484
Schaschke, Norbert, and Sommerhoff, Christian P. 2010. “Upgrading a Natural Product: Inhibition of Human beta-Tryptase by Cyclotheonamide Analogues”. CHEMMEDCHEM 5 (3): 367-370.
Schaschke, N., and Sommerhoff, C. P. (2010). Upgrading a Natural Product: Inhibition of Human beta-Tryptase by Cyclotheonamide Analogues. CHEMMEDCHEM 5, 367-370.
Schaschke, N., & Sommerhoff, C.P., 2010. Upgrading a Natural Product: Inhibition of Human beta-Tryptase by Cyclotheonamide Analogues. CHEMMEDCHEM, 5(3), p 367-370.
N. Schaschke and C.P. Sommerhoff, “Upgrading a Natural Product: Inhibition of Human beta-Tryptase by Cyclotheonamide Analogues”, CHEMMEDCHEM, vol. 5, 2010, pp. 367-370.
Schaschke, N., Sommerhoff, C.P.: Upgrading a Natural Product: Inhibition of Human beta-Tryptase by Cyclotheonamide Analogues. CHEMMEDCHEM. 5, 367-370 (2010).
Schaschke, Norbert, and Sommerhoff, Christian P. “Upgrading a Natural Product: Inhibition of Human beta-Tryptase by Cyclotheonamide Analogues”. CHEMMEDCHEM 5.3 (2010): 367-370.

5 Zitationen in Europe PMC

Daten bereitgestellt von Europe PubMed Central.

Marine Sponges as a Drug Treasure.
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Synthesis and stereochemical analysis of β-nitromethane substituted γ-amino acids and peptides.
Ganesh Kumar M, Mali SM, Gopi HN., Org Biomol Chem 11(5), 2013
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A new approach to inhibit human β-tryptase by protein surface binding of four-armed peptide ligands with two different sets of arms.
Jiang QQ, Bartsch L, Sicking W, Wich PR, Heider D, Hoffmann D, Schmuck C., Org Biomol Chem 11(10), 2013
PMID: 23358683
Synthesis of α, β-unsaturated γ-amino esters with unprecedented high (E)-stereoselectivity and their conformational analysis in peptides.
Mali SM, Bandyopadhyay A, Jadhav SV, Kumar MG, Gopi HN., Org Biomol Chem 9(19), 2011
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The arginine mimicking β-amino acid β³hPhe(3-H₂N-CH₂) as S1 ligand in cyclotheonamide-based β-tryptase inhibitors.
Janke D, Sommerhoff CP, Schaschke N., Bioorg Med Chem 19(23), 2011
PMID: 22047802

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