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21 Publikationen

2018 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 2920953
Novel unit B cryptophycin analogues as payloads for targeted therapy
Figueras Agustí E, Borbély AN, Ismail M, Frese M, Sewald N (2018)
BEILSTEIN JOURNAL OF ORGANIC CHEMISTRY 14: 1281-1286.
PUB | DOI | WoS | PubMed | Europe PMC
 
2018 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 2921235
Characterization of the Actinonin Biosynthetic Gene Cluster
Wolf F, Leipoldt F, Kulik A, Wibberg D, Kalinowski J, Kaysser L (2018)
CHEMBIOCHEM 19(11): 1189-1195.
PUB | DOI | WoS | PubMed | Europe PMC
 
2017 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 2911994
Biosynthesis of the beta-Lactone Proteasome Inhibitors Belactosin and Cystargolide
Wolf F, Bauer JS, Bendel TM, Kulik A, Kalinowski J, Gross H, Kaysser L (2017)
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 56(23): 6665-6668.
PUB | DOI | WoS | PubMed | Europe PMC
 
2017 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 2910347
Crystal structures, binding interactions, and ADME evaluation of brain penetrant N-substituted indazole-5-carboxamides as subnanomolar, selective monoamine oxidase B and dual MAO-A/B inhibitors
Tzvetkov NT, Stammler H-G, Neumann B, Hristova S, Antonov L, Gastreich M (2017)
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 127: 470-492.
PUB | DOI | WoS | PubMed | Europe PMC
 
2017 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 2915073
Tautomerism of N-(3,4-dichloropheny1)-1H-indazole-5-carboxamide - A new selective, highly potent and reversible MAO-B inhibitor
Tzvetkov NT, Stammler H-G, Antonov L (2017)
JOURNAL OF MOLECULAR STRUCTURE 1149: 273-281.
PUB | DOI | WoS
 
2017 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 2917176
Structure-Activity Relationship of Propargylamine-Based HDAC Inhibitors
Wünsch M, Senger J, Schultheisz P, Schwarzbich S, Schmidtkunz K, Michalek C, Klaß M, Goskowitz S, Borchert P, Praetorius L, Sippl W, et al. (2017)
CHEMMEDCHEM 12(24): 2044-2053.
PUB | DOI | WoS | PubMed | Europe PMC
 
2014 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 2684340
Harnessing the Evolvability of Tricyclic Microviridins To Dissect Protease-Inhibitor Interactions
Weiz AR, Ishida K, Quitterer F, Meyer S, Kehr J-C, Müller K, Groll M, Hertweck C, Dittmann E (2014)
Angewandte Chemie International Edition 53(14): 3735-3738.
PUB | DOI | WoS | PubMed | Europe PMC
 
2013 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 2613022
Conformational Properties of Secondary Amino Acids: Replacement of Pipecolic Acid by N-Methyl-L-alanine in Efrapeptin C
Konar AD, Vass E, Hollosi M, Majer Z, Grueber G, Frese K, Sewald N (2013)
Chemistry & Biodiversity 10(5): 942-951.
PUB | DOI | WoS | PubMed | Europe PMC
 
2012 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 2499381
Synthesis and conformational analysis of efrapeptins
Weigelt S, Huber T, Hofmann F, Jost M, Ritzefeld M, Luy B, Freudenberger C, Majer Z, Vass E, Greie J-C, Panella L, et al. (2012)
Chem. Eur. J. 18(2): 478-487.
PUB | DOI | WoS | PubMed | Europe PMC
 
2010 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 2576765
Human peritoneal macrophages from ascitic fluid can be infected by a broad range of HIV-1 isolates
Chang TL, Klepper A, Ding J, Garber J, Rapista A, Mosoian A, Hübner W, Gutierrez J, Walewski J, Abergel J, Schiano T, et al. (2010)
Journal of acquired immune deficiency syndromes (1999) 53(3): 292-302.
PUB | DOI | WoS | PubMed | Europe PMC
 
2009 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1588884
Cost Effectiveness of Exemestane versus Tamoxifen in Post-Menopausal Women with Early Breast Cancer in Germany
Braun S, Mittendorf T, Menschik T, Greiner W, von der Schulenburg J-M (2009)
BREAST CARE 4(6): 389-396.
PUB | DOI | WoS | PubMed | Europe PMC
 
2008 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 2403715
Inhibition of cathepsin L by epoxysuccinyl peptides simultaneously addressing active-site and remote-site regions
Schaschke N, Assfalg-Machleidt I, Machleidt W (2008)
CHEMBIOCHEM 9(11): 1721-1724.
PUB | DOI | WoS | PubMed | Europe PMC
 
2008 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1585817
Pentapeptides containing two dehydrophenylalanine residues - synthesis, structural studies and evaluation of their activity towards cathepsin C
Latajka R, Jewginski M, Makowski M, Paweiczak M, Huber T, Sewald N, Kafarski P (2008)
JOURNAL OF PEPTIDE SCIENCE 14(10): 1084-1095.
PUB | DOI | WoS | PubMed | Europe PMC
 
2007 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 2403747
Mast cell tryptase beta as a target in allergic inflammation: An evolving story
Sommerhoff CP, Schaschke N (2007)
CURRENT PHARMACEUTICAL DESIGN 13(3): 313-332.
PUB | DOI | WoS | PubMed | Europe PMC
 
2007 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1927872
Cdc42 and phosphoinositide 3-kinase drive Rac-mediated actin polymerization downstream of c-Met in distinct and common pathways
Bosse T, Ehinger J, Czuchra A, Benesch S, Steffen A, Wu X, Schloen K, Niemann H, Scita G, Stradal TE, Brakebusch C, et al. (2007)
Mol Cell Biol 27(19): 6615-6628.
PUB | DOI | WoS | PubMed | Europe PMC
 
2006 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1601428
N-hydroxyurea as zinc binding group in matrix metalloproteinase inhibition: Mode of binding in a complex with MMP-8
Campestre C, Agamennone M, Tortorella P, Preziuso S, Biasone A, Gavuzzo E, Pochetti G, Mazza F, Hiller O, Tschesche H, Consalvi V, et al. (2006)
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 16(1): 20-24.
PUB | DOI | WoS | PubMed | Europe PMC
 
2004 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1608728
Catalytic- and ecto-domains of membrane type 1-matrix metalloproteinase have similar inhibition profiles but distinct endopeptidase activities
Hurst DR, Schwartz MA, Ghaffari MA, Jin YH, Tschesche H, Fields GB, Sang QXA (2004)
BIOCHEMICAL JOURNAL 377: 775-779.
PUB | DOI | WoS | PubMed | Europe PMC
 
2003 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1609536
Affinity-based tagging of protein families with reversible inhibitors: A concept for functional proteomics
Hagenstein MC, Mussgnug JH, Lotte K, Plessow R, Brockhinke A, Kruse O, Sewald N (2003)
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION 42(45): 5635-5638.
PUB | DOI | WoS | PubMed | Europe PMC
 
2002 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1613937 PUB | DOI | WoS | PubMed | Europe PMC
 
2000 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1619233
Highly potent inhibitors of human cathepsin L identified by screening combinatorial pentapeptide amide collections
Brinker A, Weber E, Stoll D, Voigt J, Muller A, Sewald N, Jung G, Wiesmuller KH, Bohley P (2000)
EUROPEAN JOURNAL OF BIOCHEMISTRY 267(16): 5085-5092.
PUB | DOI | WoS | PubMed | Europe PMC
 

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