The constrained amino acid beta-Acc confers potency and selectivity to integrin ligands

Urman S, Gaus K, Yang Y, Strijowski U, Sewald N, De Pol S, Reiser O (2007)
Angewandte Chemie International Edition 46(21): 3976-3978.

Zeitschriftenaufsatz | Veröffentlicht | Englisch
 
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Autor*in
Urman, Sylwia; Gaus, Katharina; Yang, Yi; Strijowski, Ulf; Sewald, NorbertUniBi ; De Pol, Silvia; Reiser, Oliver
Stichworte
amino acids; integrins; peptides; structure-activity relationships; conformational analysis
Erscheinungsjahr
2007
Zeitschriftentitel
Angewandte Chemie International Edition
Band
46
Ausgabe
21
Seite(n)
3976-3978
ISSN
1433-7851
eISSN
1521-3773
Page URI
https://pub.uni-bielefeld.de/record/1593721

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Urman S, Gaus K, Yang Y, et al. The constrained amino acid beta-Acc confers potency and selectivity to integrin ligands. Angewandte Chemie International Edition. 2007;46(21):3976-3978.
Urman, S., Gaus, K., Yang, Y., Strijowski, U., Sewald, N., De Pol, S., & Reiser, O. (2007). The constrained amino acid beta-Acc confers potency and selectivity to integrin ligands. Angewandte Chemie International Edition, 46(21), 3976-3978. https://doi.org/10.1002/anie.200605248
Urman, Sylwia, Gaus, Katharina, Yang, Yi, Strijowski, Ulf, Sewald, Norbert, De Pol, Silvia, and Reiser, Oliver. 2007. “The constrained amino acid beta-Acc confers potency and selectivity to integrin ligands”. Angewandte Chemie International Edition 46 (21): 3976-3978.
Urman, S., Gaus, K., Yang, Y., Strijowski, U., Sewald, N., De Pol, S., and Reiser, O. (2007). The constrained amino acid beta-Acc confers potency and selectivity to integrin ligands. Angewandte Chemie International Edition 46, 3976-3978.
Urman, S., et al., 2007. The constrained amino acid beta-Acc confers potency and selectivity to integrin ligands. Angewandte Chemie International Edition, 46(21), p 3976-3978.
S. Urman, et al., “The constrained amino acid beta-Acc confers potency and selectivity to integrin ligands”, Angewandte Chemie International Edition, vol. 46, 2007, pp. 3976-3978.
Urman, S., Gaus, K., Yang, Y., Strijowski, U., Sewald, N., De Pol, S., Reiser, O.: The constrained amino acid beta-Acc confers potency and selectivity to integrin ligands. Angewandte Chemie International Edition. 46, 3976-3978 (2007).
Urman, Sylwia, Gaus, Katharina, Yang, Yi, Strijowski, Ulf, Sewald, Norbert, De Pol, Silvia, and Reiser, Oliver. “The constrained amino acid beta-Acc confers potency and selectivity to integrin ligands”. Angewandte Chemie International Edition 46.21 (2007): 3976-3978.

20 Zitationen in Europe PMC

Daten bereitgestellt von Europe PubMed Central.

Synthesis and Biological Evaluation of RGD⁻Cryptophycin Conjugates for Targeted Drug Delivery.
Borbély A, Figueras E, Martins A, Esposito S, Auciello G, Monteagudo E, Di Marco A, Summa V, Cordella P, Perego R, Kemker I, Frese M, Gallinari P, Steinkühler C, Sewald N., Pharmaceutics 11(4), 2019
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PMID: 24706601
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Lesma G, Salvadori S, Airaghi F, Bojnik E, Borsodi A, Recca T, Sacchetti A, Balboni G, Silvani A., Mol Divers 17(1), 2013
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PMID: 21915696
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Cyclic RGD β-lactam peptidomimetics induce differential gene expression in human endothelial cells.
Aizpurua JM, Ganboa JI, Palomo C, Loinaz I, Oyarbide J, Fernandez X, Balentová E, Fratila RM, Jiménez A, Miranda JI, Laso A, Avila S, Castrillo JL., Chembiochem 12(3), 2011
PMID: 21290542
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Pilsl LK, Reiser O., Amino Acids 41(3), 2011
PMID: 21462000
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Tolomelli A, Gentilucci L, Mosconi E, Viola A, Dattoli SD, Baiula M, Spampinato S, Belvisi L, Civera M., ChemMedChem 6(12), 2011
PMID: 21953988
Synthesis and biochemical evaluation of a cyclic RGD oxorhenium complex as new ligand of alphaVbeta3 integrin.
Aufort M, Gonera M, Chaignon N, Le Clainche L, Dugave C., Eur J Med Chem 44(9), 2009
PMID: 19303174
Cyclic RGD-peptidomimetics containing bifunctional diketopiperazine scaffolds as new potent integrin ligands.
da Ressurreição AS, Vidu A, Civera M, Belvisi L, Potenza D, Manzoni L, Ongeri S, Gennari C, Piarulli U., Chemistry 15(45), 2009
PMID: 19830748
Synthesis, SAR and in vitro evaluation of new cyclic Arg-Gly-Asp pseudopentapeptides containing a s-cis peptide bond as integrin alphavbeta3 and alphavbeta5 ligands.
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PMID: 18343671
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