Bivalent inhibition of beta-tryptase: Distance scan of neighboring subunits by dibasic inhibitors

Schaschke N, Dominik A, Matschiner G, Sommerhoff CP (2002)
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 12(6): 985-988.

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BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
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Schaschke N, Dominik A, Matschiner G, Sommerhoff CP. Bivalent inhibition of beta-tryptase: Distance scan of neighboring subunits by dibasic inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 2002;12(6):985-988.
Schaschke, N., Dominik, A., Matschiner, G., & Sommerhoff, C. P. (2002). Bivalent inhibition of beta-tryptase: Distance scan of neighboring subunits by dibasic inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 12(6), 985-988. doi:10.1016/S0960-894X(02)00063-X
Schaschke, N., Dominik, A., Matschiner, G., and Sommerhoff, C. P. (2002). Bivalent inhibition of beta-tryptase: Distance scan of neighboring subunits by dibasic inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 12, 985-988.
Schaschke, N., et al., 2002. Bivalent inhibition of beta-tryptase: Distance scan of neighboring subunits by dibasic inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 12(6), p 985-988.
N. Schaschke, et al., “Bivalent inhibition of beta-tryptase: Distance scan of neighboring subunits by dibasic inhibitors”, BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 12, 2002, pp. 985-988.
Schaschke, N., Dominik, A., Matschiner, G., Sommerhoff, C.P.: Bivalent inhibition of beta-tryptase: Distance scan of neighboring subunits by dibasic inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 12, 985-988 (2002).
Schaschke, Norbert, Dominik, A, Matschiner, G, and Sommerhoff, CP. “Bivalent inhibition of beta-tryptase: Distance scan of neighboring subunits by dibasic inhibitors”. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 12.6 (2002): 985-988.

11 Zitationen in Europe PMC

Daten bereitgestellt von Europe PubMed Central.

A new approach to inhibit human β-tryptase by protein surface binding of four-armed peptide ligands with two different sets of arms.
Jiang QQ, Bartsch L, Sicking W, Wich PR, Heider D, Hoffmann D, Schmuck C., Org Biomol Chem 11(10), 2013
PMID: 23358683
Engineered cystine knot miniproteins as potent inhibitors of human mast cell tryptase beta.
Sommerhoff CP, Avrutina O, Schmoldt HU, Gabrijelcic-Geiger D, Diederichsen U, Kolmar H., J Mol Biol 395(1), 2010
PMID: 19852971
Biology of mast cell tryptase. An inflammatory mediator.
Hallgren J, Pejler G., FEBS J 273(9), 2006
PMID: 16640553
Affinity chromatography of tryptases: design, synthesis and characterization of a novel matrix-bound bivalent inhibitor.
Schaschke N, Gabrijelcic-Geiger D, Dominik A, Sommerhoff CP., Chembiochem 6(1), 2005
PMID: 15593113
Combinatorial approaches towards the discovery of new tryptase inhibitors.
del Fresno M, Fernández-Forner D, Miralpeix M, Segarra V, Ryder H, Royo M, Albericio F., Bioorg Med Chem Lett 15(6), 2005
PMID: 15745817
Design of bivalent ligands using hydrogen bond linkers: synthesis and evaluation of inhibitors for human beta-tryptase.
Vaz RJ, Gao Z, Pribish J, Chen X, Levell J, Davis L, Albert E, Brollo M, Ugolini A, Cramer DM, Cairns J, Sides K, Liu F, Kwong J, Kang J, Rebello S, Elliot M, Lim H, Chellaraj V, Singleton RW, Li Y., Bioorg Med Chem Lett 14(24), 2004
PMID: 15546728
Potent bivalent inhibition of human tryptase-beta by a synthetic inhibitor.
Selwood T, Elrod KC, Schechter NM., Biol Chem 384(12), 2003
PMID: 14719803

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