Integrin alpha(5)beta(1) ligands: Biological evaluation and conformational analysis

Zimmermann D, Guthohrlein EW, Malesevic M, Sewald K, Wobbe L, Heggemann C, Sewald N (2005)
CHEMBIOCHEM 6(2): 272-276.

Journal Article | Published | English

No fulltext has been uploaded

Author
; ; ; ; ; ;
Publishing Year
ISSN
PUB-ID

Cite this

Zimmermann D, Guthohrlein EW, Malesevic M, et al. Integrin alpha(5)beta(1) ligands: Biological evaluation and conformational analysis. CHEMBIOCHEM. 2005;6(2):272-276.
Zimmermann, D., Guthohrlein, E. W., Malesevic, M., Sewald, K., Wobbe, L., Heggemann, C., & Sewald, N. (2005). Integrin alpha(5)beta(1) ligands: Biological evaluation and conformational analysis. CHEMBIOCHEM, 6(2), 272-276.
Zimmermann, D., Guthohrlein, E. W., Malesevic, M., Sewald, K., Wobbe, L., Heggemann, C., and Sewald, N. (2005). Integrin alpha(5)beta(1) ligands: Biological evaluation and conformational analysis. CHEMBIOCHEM 6, 272-276.
Zimmermann, D., et al., 2005. Integrin alpha(5)beta(1) ligands: Biological evaluation and conformational analysis. CHEMBIOCHEM, 6(2), p 272-276.
D. Zimmermann, et al., “Integrin alpha(5)beta(1) ligands: Biological evaluation and conformational analysis”, CHEMBIOCHEM, vol. 6, 2005, pp. 272-276.
Zimmermann, D., Guthohrlein, E.W., Malesevic, M., Sewald, K., Wobbe, L., Heggemann, C., Sewald, N.: Integrin alpha(5)beta(1) ligands: Biological evaluation and conformational analysis. CHEMBIOCHEM. 6, 272-276 (2005).
Zimmermann, D, Guthohrlein, EW, Malesevic, M, Sewald, K, Wobbe, Lutz, Heggemann, C, and Sewald, Norbert. “Integrin alpha(5)beta(1) ligands: Biological evaluation and conformational analysis”. CHEMBIOCHEM 6.2 (2005): 272-276.
This data publication is cited in the following publications:
This publication cites the following data publications:

11 Citations in Europe PMC

Data provided by Europe PubMed Central.

The integrin ligand c(RGDf(NMe)Nal) reduces neointimal hyperplasia in a polymer-free drug-eluting stent system.
Rechenmacher F, Steigerwald K, Laufer B, Neubauer S, Kapp TG, Li L, Mas-Moruno C, Joner M, Kessler H., ChemMedChem 9(7), 2014
PMID: 24706601
HUVEC cell affinity evaluation and integrin-mediated mechanism study on PHSRN-modified polymer.
Liu Y, Wang W, Wang J, Yuan Z, Tang S, Liu M, Tang H., Colloids Surf B Biointerfaces 84(1), 2011
PMID: 21216133
Conformational control of integrin-subtype selectivity in isoDGR peptide motifs: a biological switch.
Frank AO, Otto E, Mas-Moruno C, Schiller HB, Marinelli L, Cosconati S, Bochen A, Vossmeyer D, Zahn G, Stragies R, Novellino E, Kessler H., Angew. Chem. Int. Ed. Engl. 49(48), 2010
PMID: 20957712
Helicobacter pylori type IV secretion apparatus exploits beta1 integrin in a novel RGD-independent manner.
Jimenez-Soto LF, Kutter S, Sewald X, Ertl C, Weiss E, Kapp U, Rohde M, Pirch T, Jung K, Retta SF, Terradot L, Fischer W, Haas R., PLoS Pathog. 5(12), 2009
PMID: 19997503
Conformational consequences of regio- and stereoselective disulfide bridge oxidation in a cyclic peptide.
Malesevic M, Jahreis G, Wawra S, Fischer G, Lucke C., Chembiochem 9(1), 2008
PMID: 18072227
Helicobacter exploits integrin for type IV secretion and kinase activation.
Kwok T, Zabler D, Urman S, Rohde M, Hartig R, Wessler S, Misselwitz R, Berger J, Sewald N, Konig W, Backert S., Nature 449(7164), 2007
PMID: 17943123
Synthesis and biological evaluation of non-peptide alpha(v)beta(3)/alpha(5)beta(1) integrin dual antagonists containing 5,6-dihydropyridin-2-one scaffolds.
Benfatti F, Cardillo G, Fabbroni S, Galzerano P, Gentilucci L, Juris R, Tolomelli A, Baiula M, Sparta A, Spampinato S., Bioorg. Med. Chem. 15(23), 2007
PMID: 17869121
Synthesis, and structural and biological studies of efrapeptin C analogues.
Jost M, Weigelt S, Huber T, Majer Z, Greie JC, Altendorf K, Sewald N., Chem. Biodivers. 4(6), 2007
PMID: 17589859
Probing integrin selectivity: rational design of highly active and selective ligands for the alpha5beta1 and alphavbeta3 integrin receptor.
Heckmann D, Meyer A, Marinelli L, Zahn G, Stragies R, Kessler H., Angew. Chem. Int. Ed. Engl. 46(19), 2007
PMID: 17394271
The constrained amino acid beta-Acc confers potency and selectivity to integrin ligands.
Urman S, Gaus K, Yang Y, Strijowski U, Sewald N, De Pol S, Reiser O., Angew. Chem. Int. Ed. Engl. 46(21), 2007
PMID: 17394270
Survey of the year 2005 commercial optical biosensor literature.
Rich RL, Myszka DG., J. Mol. Recognit. 19(6), 2006
PMID: 17125150

24 References

Data provided by Europe PubMed Central.


cardarelli, 1996

müller, lett pept sci 4(), 1997

mould, j biol chem 270(), 1995

nath, j cell biol 112(), 1999

haubner, 1994

xu, j biol chem 275(), 2000

vella, j biol chem 278(), 2003

pfaff, j biol chem 269(), 1994
Development and application of surface plasmon resonance-based biosensors for the detection of cell-ligand interactions.
Quinn JG, O'Neill S, Doyle A, McAtamney C, Diamond D, MacCraith BD, O'Kennedy R., Anal. Biochem. 281(2), 2000
PMID: 10870828
Kinetic analysis of the interaction between HIV-1 protease and inhibitors using optical biosensor technology.
Markgren PO, Hamalainen M, Danielson UH., Anal. Biochem. 279(1), 2000
PMID: 10683232
A regulated interaction between alpha5beta1 integrin and osteopontin.
Barry ST, Ludbrook SB, Murrison E, Horgan CM., Biochem. Biophys. Res. Commun. 267(3), 2000
PMID: 10673366
Are β-Amino Acids γ-Turn Mimetics? Exploring A New Design Principle for Bioactive Cyclopeptides
Schumann, Journal of the American Chemical Society 122(48), 2000
Complex formation of platelet membrane glycoproteins IIb and IIIa with fibrinogen.
Nachman RL, Leung LL., J. Clin. Invest. 69(2), 1982
PMID: 6460044
Integrin Signaling and Matrix Assembly
Ruoslahti, Tumor Biology 17(2), 1996
BIAcore for macromolecular interaction.
Fivash M, Towler EM, Fisher RJ., Curr. Opin. Biotechnol. 9(1), 1998
PMID: 9503595
Receptor-bound conformation of an alpha(5)beta(1) integrin antagonist by (15)N-edited 2D transferred nuclear overhauser effects.
Zhang L, Mattern RH, Malaney TI, Pierschbacher MD, Goodman M., J. Am. Chem. Soc. 124(12), 2002
PMID: 11902863
MOLSCRIPT: a program to produce both detailed and schematic plots of protein structures
Kraulis, Journal of Applied Crystallography 24(5), 1991
RGD and other recognition sequences for integrins.
Ruoslahti E., Annu. Rev. Cell Dev. Biol. 12(), 1996
PMID: 8970741
Stereoisomeric Peptide Libraries and Peptidomimetics for Designing Selective Inhibitors of theαvβ3 Integrin for a New Cancer Therapy
Haubner, Angewandte Chemie International Edition in English 36(1314), 1997
Methods for analysis of the integrin ligand binding event.
Smith JW., Methods Cell Biol. 69(), 2002
PMID: 12070996
Stereoisomere Peptid-Bibliotheken und Peptidmimetika zum Design von selektiven Inhibitoren des αv β3-Integrins für eine neuartige Krebstherapie
Haubner, Angewandte Chemie 109(13-14), 1997

Export

0 Marked Publications

Open Data PUB

Web of Science

View record in Web of Science®

Sources

PMID: 15645521
PubMed | Europe PMC

Search this title in

Google Scholar