32 Publikationen

Alle markieren

  • [32]
    2001 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1617209
    Schroder, J, Wenzel, Herbert, Stammler, Hans-Georg, Stammler, A, Neumann, B, and Tschesche, Harald. 2001. “Novel heterocyclic inhibitors of matrix metalloproteinases: three 6H-1,3,4-thiadiazines”. ACTA CRYSTALLOGRAPHICA SECTION C-CRYSTAL STRUCTURE COMMUNICATIONS 57 (5): 593-596.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [31]
    2001 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1616195
    Schröder, J., Henke, A, Wenzel, Herbert, Brandstetter, H, Stammler, Hans-Georg, Stammler, A, Pfeiffer, WD, and Tschesche, Harald. 2001. “Structure-based design and synthesis of potent matrix metalloproteinase inhibitors derived from a 6H-1,3,4-thiadiazine scaffold”. JOURNAL OF MEDICINAL CHEMISTRY 44 (20): 3231-3243.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [30]
    1998 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1624672
    Krumme, D, Wenzel, Herbert, and Tschesche, Harald. 1998. “Hydroxamate derivatives of substrate-analogous peptides containing aminomalonic acid are potent inhibitors of matrix metalloproteinases”. FEBS LETTERS 436 (2): 209-212.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [29]
    1997 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1628000
    Brinkmann, T, Korfer, R, Wenzel, Herbert, Tschesche, Harald, and Kleesiek, Knut. 1997. “Strong crossreaction of human anti-aprotinin antibodies from heart transplant patient with [Arg(15)]aprotinin”. IMMUNOPHARMACOLOGY 35 (3): 221-228.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [28]
    1995 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1641415
    WACHTFOGEL, YT, HACK, CE, NUIJENS, JH, KETTNER, C, REILLY, TM, KNABB, RM, BISCHOFF, R, et al. 1995. “SELECTIVE KALLIKREIN INHIBITORS ALTER HUMAN NEUTROPHIL ELASTASE RELEASE DURING EXTRACORPOREAL-CIRCULATION”. AMERICAN JOURNAL OF PHYSIOLOGY-HEART AND CIRCULATORY PHYSIOLOGY 268 (3): H1352-H1357.
    PUB | DOI | WoS
     
  • [27]
    1994 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1642944
    GROEGER, C, Wenzel, Herbert, and Tschesche, Harald. 1994. “BPTI BACKBONE VARIANTS AND IMPLICATIONS FOR INHIBITORY ACTIVITY”. INTERNATIONAL JOURNAL OF PEPTIDE AND PROTEIN RESEARCH 44 (2): 166-172.
    PUB | WoS | PubMed | Europe PMC
     
  • [26]
    1993 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1645607
    GROEGER, C, Wenzel, Herbert, and Tschesche, Harald. 1993. “THE IMPORTANCE OF THE RIGIDITY OF THE PEPTIDE BACKBONE FOR THE INHIBITORY PROPERTIES OF BPTI DEMONSTRATED BY SEMISYNTHETIC STRUCTURAL VARIANTS”. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH 32 (6): 898-900.
    PUB | DOI | WoS
     
  • [25]
    1991 | Konferenzbeitrag | Veröffentlicht | PUB-ID: 1629600
    Tschesche, Harald, Groeger, C., and Wenzel, Herbert. 1991. “ENZYMATIC FRAGMENT SUBSTITUTION AS A TOOL IN PROTEIN DESIGN”. In Emerg Med J, 50:S175-S180. BIOMEDICA BIOCHIMICA ACTA. AKADEMIE VERLAG GMBH.
    PUB | WoS | PubMed | Europe PMC
     
  • [24]
    1991 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1649242
    GROEGER, C, Wenzel, Herbert, and Tschesche, Harald. 1991. “CHEMICAL SEMISYNTHESIS OF APROTININ HOMOLOGS AND DERIVATIVES MUTATED IN P' POSITIONS”. JOURNAL OF PROTEIN CHEMISTRY 10 (5): 527-533.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [23]
    1991 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1649962
    GROEGER, C, Wenzel, Herbert, and Tschesche, Harald. 1991. “ENZYMATIC SEMISYNTHESIS OF APROTININ HOMOLOGS MUTATED IN P' POSITIONS”. JOURNAL OF PROTEIN CHEMISTRY 10 (2): 245-251.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [22]
    1990 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1650922
    Wenzel, Herbert, FELDMANN, A, ENGELBRECHT, S, and Tschesche, Harald. 1990. “ACTIVATION OF THE HUMAN-LEUKOCYTE PROTEINASES ELASTASE AND CATHEPSIN-G BY VARIOUS SURFACTANTS”. BIOLOGICAL CHEMISTRY HOPPE-SEYLER 371 (2): 721-724.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [21]
    1989 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1652842
    MEHLICH, A, BECKMANN, J, Wenzel, Herbert, and Tschesche, Harald. 1989. “SEMISYNTHETIC APROTININ DERIVATIVES WITH SPECIFIC ALTERATIONS AT THE REACTIVE-SITE PEPTIDE-BOND CAN BE USED TO STUDY STRUCTURE-FUNCTION-RELATIONSHIPS”. BIOCHIMICA ET BIOPHYSICA ACTA 996 (1-2): 23-29.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [20]
    1989 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1652670
    SIEKMANN, J, BECKMANN, J, MEHLICH, A, Wenzel, Herbert, Tschesche, Harald, SCHNABEL, E, and MULLERESTERL, W. 1989. “IMMUNOLOGICAL CHARACTERIZATION OF NATURAL AND SEMISYNTHETIC APROTININ VARIANTS”. BIOLOGICAL CHEMISTRY HOPPE-SEYLER 370 (2): 677-682.
    PUB | DOI | WoS
     
  • [19]
    1989 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1653324
    BECKMANN, J, MEHLICH, A, SCHRODER, W, Wenzel, Herbert, and Tschesche, Harald. 1989. “SEMISYNTHESIS OF ARG-15-APROTININ, GLU-15-APROTININ, MET-15-APROTININ, AND NLE15-APROTININ INVOLVING ENZYMATIC PEPTIDE-BOND RESYNTHESIS”. JOURNAL OF PROTEIN CHEMISTRY 8 (1): 101-113.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [18]
    1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1653441
    MEHLICH, A, BECKMANN, J, Wenzel, Herbert, and Tschesche, Harald. 1988. “APROTININ DERIVATIVES WITH CHROMOPHORIC LEAVING GROUPS CAN BE USED AS HIGHLY SELECTIVE ACTIVE-SITE TITRANTS FOR SERINE PROTEINASES AND PERMIT THE DETERMINATION OF KINETIC CONSTANTS OF ENZYME-INHIBITOR COMPLEXES”. BIOCHIMICA ET BIOPHYSICA ACTA 957 (3): 420-429.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [17]
    1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1653768
    BECKMANN, J, MEHLICH, A, SCHRODER, W, Wenzel, Herbert, and Tschesche, Harald. 1988. “PREPARATION OF CHEMICALLY MUTATED APROTININ HOMOLOGS BY SEMISYNTHESIS - P1 SUBSTITUTIONS CHANGE INHIBITORY SPECIFICITY”. EUROPEAN JOURNAL OF BIOCHEMISTRY 176 (3): 675-682.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [16]
    1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1654061
    SCHNABEL, E, REINHARDT, G, SCHRODER, W, Tschesche, Harald, Wenzel, Herbert, and MEHLICH, A. 1988. “ENZYMATIC RESYNTHESIS OF THE REACTIVE SITE BOND IN THE MODIFIED APROTININ DERIVATIVES [SECO-15/16]APROTININ AND [DI-SECO-15/16,39/40]APROTININ”. BIOLOGICAL CHEMISTRY HOPPE-SEYLER 369 (1): 461-468.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [15]
    1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1654439
    SIEKMANN, J, Wenzel, Herbert, SCHRODER, W, and Tschesche, Harald. 1988. “CHARACTERIZATION AND SEQUENCE DETERMINATION OF 6 APROTININ HOMOLOGS FROM BOVINE LUNGS”. BIOLOGICAL CHEMISTRY HOPPE-SEYLER 369 (1): 157-164.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [14]
    1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1653623
    SIEKMANN, J, Wenzel, Herbert, MATUSZAK, E, VONGOLDAMMER, E, and Tschesche, Harald. 1988. “THE PH-DEPENDENCE OF THE EQUILIBRIUM-CONSTANT KHYD FOR THE HYDROLYSIS OF THE LYS15-ALA16 REACTIVE-SITE PEPTIDE-BOND IN BOVINE PANCREATIC TRYPSIN-INHIBITOR (APROTININ)”. JOURNAL OF PROTEIN CHEMISTRY 7 (5): 633-640.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [13]
    1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1948524
    Beckmann, J, Mehlich, A, Wenzel, Herbert, and Tschesche, Harald. 1988. “Semisynthetic inhibitors of human leukocyte elastase and their protective effect on lung elastin degradation in vitro”. Adv Exp Med Biol 240: 107-114.
    PUB | PubMed | Europe PMC
     
  • [12]
    1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1655390
    Tschesche, Harald, BECKMANN, J, MEHLICH, A, SCHNABEL, E, TRUSCHEIT, E, and Wenzel, Herbert. 1987. “SEMISYNTHETIC ENGINEERING OF PROTEINASE-INHIBITOR HOMOLOGS”. BIOCHIMICA ET BIOPHYSICA ACTA 913 (1): 97-101.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [11]
    1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1655547
    SCOTT, CF, Wenzel, Herbert, Tschesche, Harald, and COLMAN, RW. 1987. “KINETICS OF INHIBITION OF HUMAN-PLASMA KALLIKREIN BY A SITE-SPECIFIC MODIFIED INHIBITOR ARG15-APROTININ - EVALUATION USING A MICROPLATE SYSTEM AND COMPARISON WITH OTHER PROTEASES”. BLOOD 69 (5): 1431-1436.
    PUB | WoS | PubMed | Europe PMC
     
  • [10]
    1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1654700
    SIEKMANN, J, Wenzel, Herbert, SCHRODER, W, SCHUTT, H, TRUSCHEIT, E, ARENS, A, RAUENBUSCH, E, CHAZIN, WJ, WUTHRICH, K, and Tschesche, Harald. 1987. “PYROGLUTAMYL-APROTININ, A NEW APROTININ HOMOLOG FROM BOVINE LUNGS - ISOLATION, PROPERTIES, SEQUENCE-ANALYSIS AND CHARACTERIZATION USING HYDROGEN NUCLEAR MAGNETIC-RESONANCE IN SOLUTION”. BIOLOGICAL CHEMISTRY HOPPE-SEYLER 368 (2): 1589-1596.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [9]
    1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1654832
    HANKOVSZKY, OH, HIDEG, K, VONGOLDAMMER, E, MATUSZAK, E, KOLKENBROCK, H, Tschesche, Harald, and Wenzel, Herbert. 1987. “NEW NITROXIDE REAGENTS FOR THE SELECTIVE SPIN-LABELING AT THE GUANIDINO MOIETY OF ARGININE RESIDUES IN PEPTIDES AND PROTEINS”. BIOCHIMICA ET BIOPHYSICA ACTA 916 (1): 152-155.
    PUB | DOI | WoS
     
  • [8]
    1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1655347
    SCHWARZ, H, HINZ, HJ, MEHLICH, A, Tschesche, Harald, and Wenzel, Herbert. 1987. “STABILITY STUDIES ON DERIVATIVES OF THE BOVINE PANCREATIC TRYPSIN-INHIBITOR”. BIOCHEMISTRY 26 (12): 3544-3551.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [7]
    1984 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1658517
    BODE, W, WALTER, J, HUBER, R, Wenzel, Herbert, and Tschesche, Harald. 1984. “THE REFINED 2.2-A (0.22-NM) X-RAY CRYSTAL-STRUCTURE OF THE TERNARY COMPLEX FORMED BY BOVINE TRYPSINOGEN, VALINE-VALINE AND THE ARG15 ANALOG OF BOVINE PANCREATIC TRYPSIN-INHIBITOR”. EUROPEAN JOURNAL OF BIOCHEMISTRY 144 (1): 185-190.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [6]
    1982 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1660972
    ENGELBRECHT, S, PIEPER, E, MACARTNEY, HW, RAUTENBERG, W, Wenzel, Herbert, and Tschesche, Harald. 1982. “SEPARATION OF THE HUMAN-LEUKOCYTE ENZYMES ALANINE AMINOPEPTIDASE, CATHEPSIN-G, COLLAGENASE, ELASTASE AND MYELOPEROXIDASE”. HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE 363 (1): 305-316.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [5]
    1982 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1660931
    Wenzel, Herbert, Tschesche, Harald, VONGOLDAMMER, E, and NETZELMANN, U. 1982. “COMPLEX-FORMATION OF GUANIDINATED BOVINE TRYPSIN-INHIBITOR (KUNITZ) WITH TRYPSIN, CHYMOTRYPSIN AND TRYPSINOGEN AS STUDIED BY THE SPIN-LABEL TECHNIQUE”. FEBS LETTERS 140 (1): 53-57.
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [4]
    1982 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1660955
    BURKHARDT, H, MENNINGER, H, BERNER, W, Wenzel, Herbert, Tschesche, Harald, HOOS, R, and MIERAU, HD. 1982. “INHIBITION OF RHEUMATOID CARTILAGE DEGRADATION - A BIOMECHANICAL ASSAY FOR POTENTIAL ANTI-RHEUMATIC DRUGS”. AKTUELLE RHEUMATOLOGIE 7 (02): 60-62.
    PUB | DOI | WoS
     
  • [3]
    1981 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1661716
    Wenzel, Herbert, and Tschesche, Harald. 1981. “CHEMICAL MUTATION BY AMINO-ACID EXCHANGE IN THE REACTIVE SITE OF A PROTEINASE-INHIBITOR AND ALTERATION OF ITS INHIBITOR SPECIFITY”. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH 20 (3): 295-296.
    PUB | DOI | WoS
     
  • [2]
    1981 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1661674
    Wenzel, Herbert, and Tschesche, Harald. 1981. “CLEAVAGE OF PEPTIDE-4-NITROANILIDE SUBSTRATES WITH VARYING CHAIN-LENGTH BY HUMAN-LEUKOCYTE ELASTASE”. HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE 362 (6): 829-831.
    PUB | WoS | PubMed | Europe PMC
     
  • [1]
    1980 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1662186
    Wenzel, Herbert, ENGELBRECHT, S, REICH, H, MONDRY, W, and Tschesche, Harald. 1980. “SYNTHESIS AND ANALYTICAL USE OF 3-CARBOXYPROPIONYL-ALANYL-ALANYL-VALINE-4-NITROANILIDE - A SPECIFIC SUBSTRATE FOR HUMAN-LEUKOCYTE ELASTASE”. HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE 361 (2): 1413-1416.
    PUB | DOI | WoS | PubMed | Europe PMC
     

Suche

Publikationen filtern

Darstellung / Sortierung

Export / Einbettung