32 Publikationen

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  • [32]
    2001 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1617209
    Schroder, J., Wenzel, H., Stammler, H. - G., Stammler, A., Neumann, B., & Tschesche, H. (2001). Novel heterocyclic inhibitors of matrix metalloproteinases: three 6H-1,3,4-thiadiazines. ACTA CRYSTALLOGRAPHICA SECTION C-CRYSTAL STRUCTURE COMMUNICATIONS, 57(5), 593-596. https://doi.org/10.1107/S0108270101002372
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  • [31]
    2001 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1616195
    Schröder, J., Henke, A., Wenzel, H., Brandstetter, H., Stammler, H. - G., Stammler, A., Pfeiffer, W. D., et al. (2001). Structure-based design and synthesis of potent matrix metalloproteinase inhibitors derived from a 6H-1,3,4-thiadiazine scaffold. JOURNAL OF MEDICINAL CHEMISTRY, 44(20), 3231-3243. https://doi.org/10.1021/jm010887p
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  • [30]
    1998 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1624672
    Krumme, D., Wenzel, H., & Tschesche, H. (1998). Hydroxamate derivatives of substrate-analogous peptides containing aminomalonic acid are potent inhibitors of matrix metalloproteinases. FEBS LETTERS, 436(2), 209-212. https://doi.org/10.1016/S0014-5793(98)01128-4
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  • [29]
    1997 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1628000
    Brinkmann, T., Korfer, R., Wenzel, H., Tschesche, H., & Kleesiek, K. (1997). Strong crossreaction of human anti-aprotinin antibodies from heart transplant patient with [Arg(15)]aprotinin. IMMUNOPHARMACOLOGY, 35(3), 221-228. https://doi.org/10.1016/S0162-3109(96)00148-8
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  • [28]
    1995 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1641415
    WACHTFOGEL, Y. T., HACK, C. E., NUIJENS, J. H., KETTNER, C., REILLY, T. M., KNABB, R. M., BISCHOFF, R., et al. (1995). SELECTIVE KALLIKREIN INHIBITORS ALTER HUMAN NEUTROPHIL ELASTASE RELEASE DURING EXTRACORPOREAL-CIRCULATION. AMERICAN JOURNAL OF PHYSIOLOGY-HEART AND CIRCULATORY PHYSIOLOGY, 268(3), H1352-H1357. https://doi.org/10.1152/ajpheart.1995.268.3.H1352
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  • [27]
    1994 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1642944
    GROEGER, C., Wenzel, H., & Tschesche, H. (1994). BPTI BACKBONE VARIANTS AND IMPLICATIONS FOR INHIBITORY ACTIVITY. INTERNATIONAL JOURNAL OF PEPTIDE AND PROTEIN RESEARCH, 44(2), 166-172.
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  • [26]
    1993 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1645607
    GROEGER, C., Wenzel, H., & Tschesche, H. (1993). THE IMPORTANCE OF THE RIGIDITY OF THE PEPTIDE BACKBONE FOR THE INHIBITORY PROPERTIES OF BPTI DEMONSTRATED BY SEMISYNTHETIC STRUCTURAL VARIANTS. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH, 32(6), 898-900. https://doi.org/10.1002/anie.199308981
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  • [25]
    1991 | Konferenzbeitrag | Veröffentlicht | PUB-ID: 1629600
    Tschesche, H., Groeger, C., & Wenzel, H. (1991). ENZYMATIC FRAGMENT SUBSTITUTION AS A TOOL IN PROTEIN DESIGN. Emerg Med J, BIOMEDICA BIOCHIMICA ACTA, 50, S175-S180. AKADEMIE VERLAG GMBH.
    PUB | WoS | PubMed | Europe PMC
     
  • [24]
    1991 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1649242
    GROEGER, C., Wenzel, H., & Tschesche, H. (1991). CHEMICAL SEMISYNTHESIS OF APROTININ HOMOLOGS AND DERIVATIVES MUTATED IN P' POSITIONS. JOURNAL OF PROTEIN CHEMISTRY, 10(5), 527-533. https://doi.org/10.1007/BF01025481
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  • [23]
    1991 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1649962
    GROEGER, C., Wenzel, H., & Tschesche, H. (1991). ENZYMATIC SEMISYNTHESIS OF APROTININ HOMOLOGS MUTATED IN P' POSITIONS. JOURNAL OF PROTEIN CHEMISTRY, 10(2), 245-251. https://doi.org/10.1007/BF01024788
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  • [22]
    1990 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1650922
    Wenzel, H., FELDMANN, A., ENGELBRECHT, S., & Tschesche, H. (1990). ACTIVATION OF THE HUMAN-LEUKOCYTE PROTEINASES ELASTASE AND CATHEPSIN-G BY VARIOUS SURFACTANTS. BIOLOGICAL CHEMISTRY HOPPE-SEYLER, 371(2), 721-724. https://doi.org/10.1515/bchm3.1990.371.2.721
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  • [21]
    1989 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1652842
    MEHLICH, A., BECKMANN, J., Wenzel, H., & Tschesche, H. (1989). SEMISYNTHETIC APROTININ DERIVATIVES WITH SPECIFIC ALTERATIONS AT THE REACTIVE-SITE PEPTIDE-BOND CAN BE USED TO STUDY STRUCTURE-FUNCTION-RELATIONSHIPS. BIOCHIMICA ET BIOPHYSICA ACTA, 996(1-2), 23-29. https://doi.org/10.1016/0167-4838(89)90089-7
    PUB | DOI | WoS | PubMed | Europe PMC
     
  • [20]
    1989 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1652670
    SIEKMANN, J., BECKMANN, J., MEHLICH, A., Wenzel, H., Tschesche, H., SCHNABEL, E., & MULLERESTERL, W. (1989). IMMUNOLOGICAL CHARACTERIZATION OF NATURAL AND SEMISYNTHETIC APROTININ VARIANTS. BIOLOGICAL CHEMISTRY HOPPE-SEYLER, 370(2), 677-682. https://doi.org/10.1515/bchm3.1989.370.2.677
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  • [19]
    1989 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1653324
    BECKMANN, J., MEHLICH, A., SCHRODER, W., Wenzel, H., & Tschesche, H. (1989). SEMISYNTHESIS OF ARG-15-APROTININ, GLU-15-APROTININ, MET-15-APROTININ, AND NLE15-APROTININ INVOLVING ENZYMATIC PEPTIDE-BOND RESYNTHESIS. JOURNAL OF PROTEIN CHEMISTRY, 8(1), 101-113. https://doi.org/10.1007/BF01025082
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  • [18]
    1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1653441
    MEHLICH, A., BECKMANN, J., Wenzel, H., & Tschesche, H. (1988). APROTININ DERIVATIVES WITH CHROMOPHORIC LEAVING GROUPS CAN BE USED AS HIGHLY SELECTIVE ACTIVE-SITE TITRANTS FOR SERINE PROTEINASES AND PERMIT THE DETERMINATION OF KINETIC CONSTANTS OF ENZYME-INHIBITOR COMPLEXES. BIOCHIMICA ET BIOPHYSICA ACTA, 957(3), 420-429. https://doi.org/10.1016/0167-4838(88)90233-6
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  • [17]
    1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1653768
    BECKMANN, J., MEHLICH, A., SCHRODER, W., Wenzel, H., & Tschesche, H. (1988). PREPARATION OF CHEMICALLY MUTATED APROTININ HOMOLOGS BY SEMISYNTHESIS - P1 SUBSTITUTIONS CHANGE INHIBITORY SPECIFICITY. EUROPEAN JOURNAL OF BIOCHEMISTRY, 176(3), 675-682. https://doi.org/10.1111/j.1432-1033.1988.tb14330.x
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  • [16]
    1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1654061
    SCHNABEL, E., REINHARDT, G., SCHRODER, W., Tschesche, H., Wenzel, H., & MEHLICH, A. (1988). ENZYMATIC RESYNTHESIS OF THE REACTIVE SITE BOND IN THE MODIFIED APROTININ DERIVATIVES [SECO-15/16]APROTININ AND [DI-SECO-15/16,39/40]APROTININ. BIOLOGICAL CHEMISTRY HOPPE-SEYLER, 369(1), 461-468. https://doi.org/10.1515/bchm3.1988.369.1.461
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  • [15]
    1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1654439
    SIEKMANN, J., Wenzel, H., SCHRODER, W., & Tschesche, H. (1988). CHARACTERIZATION AND SEQUENCE DETERMINATION OF 6 APROTININ HOMOLOGS FROM BOVINE LUNGS. BIOLOGICAL CHEMISTRY HOPPE-SEYLER, 369(1), 157-164. https://doi.org/10.1515/bchm3.1988.369.1.157
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  • [14]
    1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1653623
    SIEKMANN, J., Wenzel, H., MATUSZAK, E., VONGOLDAMMER, E., & Tschesche, H. (1988). THE PH-DEPENDENCE OF THE EQUILIBRIUM-CONSTANT KHYD FOR THE HYDROLYSIS OF THE LYS15-ALA16 REACTIVE-SITE PEPTIDE-BOND IN BOVINE PANCREATIC TRYPSIN-INHIBITOR (APROTININ). JOURNAL OF PROTEIN CHEMISTRY, 7(5), 633-640. https://doi.org/10.1007/BF01024879
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  • [13]
    1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1948524
    Beckmann, J., Mehlich, A., Wenzel, H., & Tschesche, H. (1988). Semisynthetic inhibitors of human leukocyte elastase and their protective effect on lung elastin degradation in vitro. Adv Exp Med Biol, 240, 107-114.
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  • [12]
    1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1655390
    Tschesche, H., BECKMANN, J., MEHLICH, A., SCHNABEL, E., TRUSCHEIT, E., & Wenzel, H. (1987). SEMISYNTHETIC ENGINEERING OF PROTEINASE-INHIBITOR HOMOLOGS. BIOCHIMICA ET BIOPHYSICA ACTA, 913(1), 97-101. https://doi.org/10.1016/0167-4838(87)90238-X
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  • [11]
    1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1655547
    SCOTT, C. F., Wenzel, H., Tschesche, H., & COLMAN, R. W. (1987). KINETICS OF INHIBITION OF HUMAN-PLASMA KALLIKREIN BY A SITE-SPECIFIC MODIFIED INHIBITOR ARG15-APROTININ - EVALUATION USING A MICROPLATE SYSTEM AND COMPARISON WITH OTHER PROTEASES. BLOOD, 69(5), 1431-1436.
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  • [10]
    1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1654700
    SIEKMANN, J., Wenzel, H., SCHRODER, W., SCHUTT, H., TRUSCHEIT, E., ARENS, A., RAUENBUSCH, E., et al. (1987). PYROGLUTAMYL-APROTININ, A NEW APROTININ HOMOLOG FROM BOVINE LUNGS - ISOLATION, PROPERTIES, SEQUENCE-ANALYSIS AND CHARACTERIZATION USING HYDROGEN NUCLEAR MAGNETIC-RESONANCE IN SOLUTION. BIOLOGICAL CHEMISTRY HOPPE-SEYLER, 368(2), 1589-1596. https://doi.org/10.1515/bchm3.1987.368.2.1589
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  • [9]
    1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1654832
    HANKOVSZKY, O. H., HIDEG, K., VONGOLDAMMER, E., MATUSZAK, E., KOLKENBROCK, H., Tschesche, H., & Wenzel, H. (1987). NEW NITROXIDE REAGENTS FOR THE SELECTIVE SPIN-LABELING AT THE GUANIDINO MOIETY OF ARGININE RESIDUES IN PEPTIDES AND PROTEINS. BIOCHIMICA ET BIOPHYSICA ACTA, 916(1), 152-155. https://doi.org/10.1016/0167-4838(87)90223-8
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  • [8]
    1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1655347
    SCHWARZ, H., HINZ, H. J., MEHLICH, A., Tschesche, H., & Wenzel, H. (1987). STABILITY STUDIES ON DERIVATIVES OF THE BOVINE PANCREATIC TRYPSIN-INHIBITOR. BIOCHEMISTRY, 26(12), 3544-3551. https://doi.org/10.1021/bi00386a044
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  • [7]
    1984 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1658517
    BODE, W., WALTER, J., HUBER, R., Wenzel, H., & Tschesche, H. (1984). THE REFINED 2.2-A (0.22-NM) X-RAY CRYSTAL-STRUCTURE OF THE TERNARY COMPLEX FORMED BY BOVINE TRYPSINOGEN, VALINE-VALINE AND THE ARG15 ANALOG OF BOVINE PANCREATIC TRYPSIN-INHIBITOR. EUROPEAN JOURNAL OF BIOCHEMISTRY, 144(1), 185-190. https://doi.org/10.1111/j.1432-1033.1984.tb08447.x
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  • [6]
    1982 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1660972
    ENGELBRECHT, S., PIEPER, E., MACARTNEY, H. W., RAUTENBERG, W., Wenzel, H., & Tschesche, H. (1982). SEPARATION OF THE HUMAN-LEUKOCYTE ENZYMES ALANINE AMINOPEPTIDASE, CATHEPSIN-G, COLLAGENASE, ELASTASE AND MYELOPEROXIDASE. HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE, 363(1), 305-316. https://doi.org/10.1515/bchm2.1982.363.1.305
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  • [5]
    1982 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1660931
    Wenzel, H., Tschesche, H., VONGOLDAMMER, E., & NETZELMANN, U. (1982). COMPLEX-FORMATION OF GUANIDINATED BOVINE TRYPSIN-INHIBITOR (KUNITZ) WITH TRYPSIN, CHYMOTRYPSIN AND TRYPSINOGEN AS STUDIED BY THE SPIN-LABEL TECHNIQUE. FEBS LETTERS, 140(1), 53-57. https://doi.org/10.1016/0014-5793(82)80519-X
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  • [4]
    1982 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1660955
    BURKHARDT, H., MENNINGER, H., BERNER, W., Wenzel, H., Tschesche, H., HOOS, R., & MIERAU, H. D. (1982). INHIBITION OF RHEUMATOID CARTILAGE DEGRADATION - A BIOMECHANICAL ASSAY FOR POTENTIAL ANTI-RHEUMATIC DRUGS. AKTUELLE RHEUMATOLOGIE, 7(02), 60-62. https://doi.org/10.1055/s-2008-1051109
    PUB | DOI | WoS
     
  • [3]
    1981 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1661716
    Wenzel, H., & Tschesche, H. (1981). CHEMICAL MUTATION BY AMINO-ACID EXCHANGE IN THE REACTIVE SITE OF A PROTEINASE-INHIBITOR AND ALTERATION OF ITS INHIBITOR SPECIFITY. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH, 20(3), 295-296. https://doi.org/10.1002/anie.198102951
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  • [2]
    1981 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1661674
    Wenzel, H., & Tschesche, H. (1981). CLEAVAGE OF PEPTIDE-4-NITROANILIDE SUBSTRATES WITH VARYING CHAIN-LENGTH BY HUMAN-LEUKOCYTE ELASTASE. HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE, 362(6), 829-831.
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  • [1]
    1980 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1662186
    Wenzel, H., ENGELBRECHT, S., REICH, H., MONDRY, W., & Tschesche, H. (1980). SYNTHESIS AND ANALYTICAL USE OF 3-CARBOXYPROPIONYL-ALANYL-ALANYL-VALINE-4-NITROANILIDE - A SPECIFIC SUBSTRATE FOR HUMAN-LEUKOCYTE ELASTASE. HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE, 361(2), 1413-1416. https://doi.org/10.1515/bchm2.1980.361.2.1413
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