32 Publikationen
-
2001 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1617209J. Schroder, H. Wenzel, H. - G. Stammler, A. Stammler, B. Neumann, and H. Tschesche, “Novel heterocyclic inhibitors of matrix metalloproteinases: three 6H-1,3,4-thiadiazines”, ACTA CRYSTALLOGRAPHICA SECTION C-CRYSTAL STRUCTURE COMMUNICATIONS, 2001, 57, 593-596.PUB | DOI | WoS | PubMed | Europe PMC
-
2001 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1616195J. Schröder, A. Henke, H. Wenzel, H. Brandstetter, H. - G. Stammler, A. Stammler, W. D. Pfeiffer, and H. Tschesche, “Structure-based design and synthesis of potent matrix metalloproteinase inhibitors derived from a 6H-1,3,4-thiadiazine scaffold”, JOURNAL OF MEDICINAL CHEMISTRY, 2001, 44, 3231-3243.PUB | DOI | WoS | PubMed | Europe PMC
-
1998 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1624672D. Krumme, H. Wenzel, and H. Tschesche, “Hydroxamate derivatives of substrate-analogous peptides containing aminomalonic acid are potent inhibitors of matrix metalloproteinases”, FEBS LETTERS, 1998, 436, 209-212.PUB | DOI | WoS | PubMed | Europe PMC
-
1997 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1628000T. Brinkmann, R. Korfer, H. Wenzel, H. Tschesche, and K. Kleesiek, “Strong crossreaction of human anti-aprotinin antibodies from heart transplant patient with [Arg(15)]aprotinin”, IMMUNOPHARMACOLOGY, 1997, 35, 221-228.PUB | DOI | WoS | PubMed | Europe PMC
-
1995 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1641415Y. T. WACHTFOGEL, C. E. HACK, J. H. NUIJENS, C. KETTNER, T. M. REILLY, R. M. KNABB, R. BISCHOFF, H. Tschesche, H. Wenzel, U. KUCICH, et al., “SELECTIVE KALLIKREIN INHIBITORS ALTER HUMAN NEUTROPHIL ELASTASE RELEASE DURING EXTRACORPOREAL-CIRCULATION”, AMERICAN JOURNAL OF PHYSIOLOGY-HEART AND CIRCULATORY PHYSIOLOGY, 1995, 268, H1352-H1357.PUB | DOI | WoS
-
1994 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1642944C. GROEGER, H. Wenzel, and H. Tschesche, “BPTI BACKBONE VARIANTS AND IMPLICATIONS FOR INHIBITORY ACTIVITY”, INTERNATIONAL JOURNAL OF PEPTIDE AND PROTEIN RESEARCH, 1994, 44, 166-172.PUB | WoS | PubMed | Europe PMC
-
1993 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1645607C. GROEGER, H. Wenzel, and H. Tschesche, “THE IMPORTANCE OF THE RIGIDITY OF THE PEPTIDE BACKBONE FOR THE INHIBITORY PROPERTIES OF BPTI DEMONSTRATED BY SEMISYNTHETIC STRUCTURAL VARIANTS”, ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH, 1993, 32, 898-900.PUB | DOI | WoS
-
1991 | Konferenzbeitrag | Veröffentlicht | PUB-ID: 1629600H. Tschesche, C. Groeger, and H. Wenzel, in Emerg Med J, Akademie Verlag Gmbh, 1991, p. S175-S180.PUB | WoS | PubMed | Europe PMC
-
1991 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1649242C. GROEGER, H. Wenzel, and H. Tschesche, “CHEMICAL SEMISYNTHESIS OF APROTININ HOMOLOGS AND DERIVATIVES MUTATED IN P' POSITIONS”, JOURNAL OF PROTEIN CHEMISTRY, 1991, 10, 527-533.PUB | DOI | WoS | PubMed | Europe PMC
-
1991 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1649962C. GROEGER, H. Wenzel, and H. Tschesche, “ENZYMATIC SEMISYNTHESIS OF APROTININ HOMOLOGS MUTATED IN P' POSITIONS”, JOURNAL OF PROTEIN CHEMISTRY, 1991, 10, 245-251.PUB | DOI | WoS | PubMed | Europe PMC
-
1990 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1650922H. Wenzel, A. FELDMANN, S. ENGELBRECHT, and H. Tschesche, “ACTIVATION OF THE HUMAN-LEUKOCYTE PROTEINASES ELASTASE AND CATHEPSIN-G BY VARIOUS SURFACTANTS”, BIOLOGICAL CHEMISTRY HOPPE-SEYLER, 1990, 371, 721-724.PUB | DOI | WoS | PubMed | Europe PMC
-
1989 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1652842A. MEHLICH, J. BECKMANN, H. Wenzel, and H. Tschesche, “SEMISYNTHETIC APROTININ DERIVATIVES WITH SPECIFIC ALTERATIONS AT THE REACTIVE-SITE PEPTIDE-BOND CAN BE USED TO STUDY STRUCTURE-FUNCTION-RELATIONSHIPS”, BIOCHIMICA ET BIOPHYSICA ACTA, 1989, 996, 23-29.PUB | DOI | WoS | PubMed | Europe PMC
-
1989 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1652670J. SIEKMANN, J. BECKMANN, A. MEHLICH, H. Wenzel, H. Tschesche, E. SCHNABEL, and W. MULLERESTERL, “IMMUNOLOGICAL CHARACTERIZATION OF NATURAL AND SEMISYNTHETIC APROTININ VARIANTS”, BIOLOGICAL CHEMISTRY HOPPE-SEYLER, 1989, 370, 677-682.PUB | DOI | WoS
-
1989 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1653324J. BECKMANN, A. MEHLICH, W. SCHRODER, H. Wenzel, and H. Tschesche, “SEMISYNTHESIS OF ARG-15-APROTININ, GLU-15-APROTININ, MET-15-APROTININ, AND NLE15-APROTININ INVOLVING ENZYMATIC PEPTIDE-BOND RESYNTHESIS”, JOURNAL OF PROTEIN CHEMISTRY, 1989, 8, 101-113.PUB | DOI | WoS | PubMed | Europe PMC
-
1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1653441A. MEHLICH, J. BECKMANN, H. Wenzel, and H. Tschesche, “APROTININ DERIVATIVES WITH CHROMOPHORIC LEAVING GROUPS CAN BE USED AS HIGHLY SELECTIVE ACTIVE-SITE TITRANTS FOR SERINE PROTEINASES AND PERMIT THE DETERMINATION OF KINETIC CONSTANTS OF ENZYME-INHIBITOR COMPLEXES”, BIOCHIMICA ET BIOPHYSICA ACTA, 1988, 957, 420-429.PUB | DOI | WoS | PubMed | Europe PMC
-
1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1653768J. BECKMANN, A. MEHLICH, W. SCHRODER, H. Wenzel, and H. Tschesche, “PREPARATION OF CHEMICALLY MUTATED APROTININ HOMOLOGS BY SEMISYNTHESIS - P1 SUBSTITUTIONS CHANGE INHIBITORY SPECIFICITY”, EUROPEAN JOURNAL OF BIOCHEMISTRY, 1988, 176, 675-682.PUB | DOI | WoS | PubMed | Europe PMC
-
1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1654061E. SCHNABEL, G. REINHARDT, W. SCHRODER, H. Tschesche, H. Wenzel, and A. MEHLICH, “ENZYMATIC RESYNTHESIS OF THE REACTIVE SITE BOND IN THE MODIFIED APROTININ DERIVATIVES [SECO-15/16]APROTININ AND [DI-SECO-15/16,39/40]APROTININ”, BIOLOGICAL CHEMISTRY HOPPE-SEYLER, 1988, 369, 461-468.PUB | DOI | WoS | PubMed | Europe PMC
-
1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1654439J. SIEKMANN, H. Wenzel, W. SCHRODER, and H. Tschesche, “CHARACTERIZATION AND SEQUENCE DETERMINATION OF 6 APROTININ HOMOLOGS FROM BOVINE LUNGS”, BIOLOGICAL CHEMISTRY HOPPE-SEYLER, 1988, 369, 157-164.PUB | DOI | WoS | PubMed | Europe PMC
-
1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1653623J. SIEKMANN, H. Wenzel, E. MATUSZAK, E. VONGOLDAMMER, and H. Tschesche, “THE PH-DEPENDENCE OF THE EQUILIBRIUM-CONSTANT KHYD FOR THE HYDROLYSIS OF THE LYS15-ALA16 REACTIVE-SITE PEPTIDE-BOND IN BOVINE PANCREATIC TRYPSIN-INHIBITOR (APROTININ)”, JOURNAL OF PROTEIN CHEMISTRY, 1988, 7, 633-640.PUB | DOI | WoS | PubMed | Europe PMC
-
1988 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1948524J. Beckmann, A. Mehlich, H. Wenzel, and H. Tschesche, “Semisynthetic inhibitors of human leukocyte elastase and their protective effect on lung elastin degradation in vitro”, Adv Exp Med Biol, 1988, 240, 107-114.PUB | PubMed | Europe PMC
-
1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1655390H. Tschesche, J. BECKMANN, A. MEHLICH, E. SCHNABEL, E. TRUSCHEIT, and H. Wenzel, “SEMISYNTHETIC ENGINEERING OF PROTEINASE-INHIBITOR HOMOLOGS”, BIOCHIMICA ET BIOPHYSICA ACTA, 1987, 913, 97-101.PUB | DOI | WoS | PubMed | Europe PMC
-
1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1655547C. F. SCOTT, H. Wenzel, H. Tschesche, and R. W. COLMAN, “KINETICS OF INHIBITION OF HUMAN-PLASMA KALLIKREIN BY A SITE-SPECIFIC MODIFIED INHIBITOR ARG15-APROTININ - EVALUATION USING A MICROPLATE SYSTEM AND COMPARISON WITH OTHER PROTEASES”, BLOOD, 1987, 69, 1431-1436.PUB | WoS | PubMed | Europe PMC
-
1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1654700J. SIEKMANN, H. Wenzel, W. SCHRODER, H. SCHUTT, E. TRUSCHEIT, A. ARENS, E. RAUENBUSCH, W. J. CHAZIN, K. WUTHRICH, and H. Tschesche, “PYROGLUTAMYL-APROTININ, A NEW APROTININ HOMOLOG FROM BOVINE LUNGS - ISOLATION, PROPERTIES, SEQUENCE-ANALYSIS AND CHARACTERIZATION USING HYDROGEN NUCLEAR MAGNETIC-RESONANCE IN SOLUTION”, BIOLOGICAL CHEMISTRY HOPPE-SEYLER, 1987, 368, 1589-1596.PUB | DOI | WoS | PubMed | Europe PMC
-
1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1654832O. H. HANKOVSZKY, K. HIDEG, E. VONGOLDAMMER, E. MATUSZAK, H. KOLKENBROCK, H. Tschesche, and H. Wenzel, “NEW NITROXIDE REAGENTS FOR THE SELECTIVE SPIN-LABELING AT THE GUANIDINO MOIETY OF ARGININE RESIDUES IN PEPTIDES AND PROTEINS”, BIOCHIMICA ET BIOPHYSICA ACTA, 1987, 916, 152-155.PUB | DOI | WoS
-
1987 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1655347H. SCHWARZ, H. J. HINZ, A. MEHLICH, H. Tschesche, and H. Wenzel, “STABILITY STUDIES ON DERIVATIVES OF THE BOVINE PANCREATIC TRYPSIN-INHIBITOR”, BIOCHEMISTRY, 1987, 26, 3544-3551.PUB | DOI | WoS | PubMed | Europe PMC
-
1984 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1658517W. BODE, J. WALTER, R. HUBER, H. Wenzel, and H. Tschesche, “THE REFINED 2.2-A (0.22-NM) X-RAY CRYSTAL-STRUCTURE OF THE TERNARY COMPLEX FORMED BY BOVINE TRYPSINOGEN, VALINE-VALINE AND THE ARG15 ANALOG OF BOVINE PANCREATIC TRYPSIN-INHIBITOR”, EUROPEAN JOURNAL OF BIOCHEMISTRY, 1984, 144, 185-190.PUB | DOI | WoS | PubMed | Europe PMC
-
1982 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1660972S. ENGELBRECHT, E. PIEPER, H. W. MACARTNEY, W. RAUTENBERG, H. Wenzel, and H. Tschesche, “SEPARATION OF THE HUMAN-LEUKOCYTE ENZYMES ALANINE AMINOPEPTIDASE, CATHEPSIN-G, COLLAGENASE, ELASTASE AND MYELOPEROXIDASE”, HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE, 1982, 363, 305-316.PUB | DOI | WoS | PubMed | Europe PMC
-
1982 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1660931H. Wenzel, H. Tschesche, E. VONGOLDAMMER, and U. NETZELMANN, “COMPLEX-FORMATION OF GUANIDINATED BOVINE TRYPSIN-INHIBITOR (KUNITZ) WITH TRYPSIN, CHYMOTRYPSIN AND TRYPSINOGEN AS STUDIED BY THE SPIN-LABEL TECHNIQUE”, FEBS LETTERS, 1982, 140, 53-57.PUB | DOI | WoS | PubMed | Europe PMC
-
1982 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1660955H. BURKHARDT, H. MENNINGER, W. BERNER, H. Wenzel, H. Tschesche, R. HOOS, and H. D. MIERAU, “INHIBITION OF RHEUMATOID CARTILAGE DEGRADATION - A BIOMECHANICAL ASSAY FOR POTENTIAL ANTI-RHEUMATIC DRUGS”, AKTUELLE RHEUMATOLOGIE, 1982, 7, 60-62.PUB | DOI | WoS
-
1981 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1661716H. Wenzel, and H. Tschesche, “CHEMICAL MUTATION BY AMINO-ACID EXCHANGE IN THE REACTIVE SITE OF A PROTEINASE-INHIBITOR AND ALTERATION OF ITS INHIBITOR SPECIFITY”, ANGEWANDTE CHEMIE-INTERNATIONAL EDITION IN ENGLISH, 1981, 20, 295-296.PUB | DOI | WoS
-
1981 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1661674H. Wenzel, and H. Tschesche, “CLEAVAGE OF PEPTIDE-4-NITROANILIDE SUBSTRATES WITH VARYING CHAIN-LENGTH BY HUMAN-LEUKOCYTE ELASTASE”, HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE, 1981, 362, 829-831.PUB | WoS | PubMed | Europe PMC
-
1980 | Zeitschriftenaufsatz | Veröffentlicht | PUB-ID: 1662186H. Wenzel, S. ENGELBRECHT, H. REICH, W. MONDRY, and H. Tschesche, “SYNTHESIS AND ANALYTICAL USE OF 3-CARBOXYPROPIONYL-ALANYL-ALANYL-VALINE-4-NITROANILIDE - A SPECIFIC SUBSTRATE FOR HUMAN-LEUKOCYTE ELASTASE”, HOPPE-SEYLERS ZEITSCHRIFT FUR PHYSIOLOGISCHE CHEMIE, 1980, 361, 1413-1416.PUB | DOI | WoS | PubMed | Europe PMC